Table 3—

Pharmacokinetic properties of inhaled corticosteroids

Oral bioavailability%Protein-binding%ClearanceL·h-1VdLHalf-lifeh
BDP1587230200.1
BMP26NA120#424#2.7
BUD1188841832.8
CIC<1991522070.4
des-CIC<199396#1190#3.6−5.1
FLU78058961.6
FP<1906931814.4
MF<1<9853.53324.5
TAA2371371032.0
  • Vd: volume of distribution; BDP: beclometasone dipropionate; BMP: beclometasone monopropionate; BUD: budesonide; CIC: ciclesonide; des-CIC: desisobutyryl-CIC; FLU: flunisolide; FP: fluticasone propionate; MF: mometasone furoate; TAA: triamcinolone acetonide; NA: not available. #: apparent maximum approximation based on complete conversion of the parent compound. Data taken and collated from 21, 35, 4653.